Efficient Synthesis of 3-(Arenesulfinyl)indoles in Water

Y. Liu; Z. Y. Zhang; Y. Z. Ji; H. J. Li; Y. C. Wu

doi:10.1134/S1070428021050109

Efficient Synthesis of 3-(Arenesulfinyl)indoles in Water

Y. Liu^*
, Z. Y. Zhang
, Y. Z. Ji
, H. J. Li
, Y. C. Wu^*

^*Corresponding author for this work

Harbin Institute of Technolo-gy
Ltd.

Research output: Contribution to journal › Article › peer-review

2 Scopus citations

Abstract

Abstract: The first example of the sulfinylation of indoles with arylsulfinamides in water in the presence of trifluoroacetic acid as a promoter is described. The reaction occurs smoothly at room temperature under environmentally benign conditions without any catalyst, additive, ligand, or organic solvent. The developed sulfoxide synthetic protocol is attractive due to the use of water as the solvent and provides a novel and efficient route to a wide range of functionalized diaryl sulfoxides.

Original language	English
Pages (from-to)	831-841
Number of pages	11
Journal	Russian Journal of Organic Chemistry
Volume	57
Issue number	5
DOIs	https://doi.org/10.1134/S1070428021050109
State	Published - May 2021
Externally published	Yes

Keywords

indoles
sulfinylation reaction
trifluoroacetic acid
water

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10.1134/S1070428021050109

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title = "Efficient Synthesis of 3-(Arenesulfinyl)indoles in Water",

abstract = "Abstract: The first example of the sulfinylation of indoles with arylsulfinamides in water in the presence of trifluoroacetic acid as a promoter is described. The reaction occurs smoothly at room temperature under environmentally benign conditions without any catalyst, additive, ligand, or organic solvent. The developed sulfoxide synthetic protocol is attractive due to the use of water as the solvent and provides a novel and efficient route to a wide range of functionalized diaryl sulfoxides.",

keywords = "indoles, sulfinylation reaction, trifluoroacetic acid, water",

author = "Y. Liu and Zhang, \{Z. Y.\} and Ji, \{Y. Z.\} and Li, \{H. J.\} and Wu, \{Y. C.\}",

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year = "2021",

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doi = "10.1134/S1070428021050109",

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issn = "1070-4280",

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T1 - Efficient Synthesis of 3-(Arenesulfinyl)indoles in Water

AU - Liu, Y.

AU - Zhang, Z. Y.

AU - Ji, Y. Z.

AU - Li, H. J.

AU - Wu, Y. C.

PY - 2021/5

Y1 - 2021/5

N2 - Abstract: The first example of the sulfinylation of indoles with arylsulfinamides in water in the presence of trifluoroacetic acid as a promoter is described. The reaction occurs smoothly at room temperature under environmentally benign conditions without any catalyst, additive, ligand, or organic solvent. The developed sulfoxide synthetic protocol is attractive due to the use of water as the solvent and provides a novel and efficient route to a wide range of functionalized diaryl sulfoxides.

AB - Abstract: The first example of the sulfinylation of indoles with arylsulfinamides in water in the presence of trifluoroacetic acid as a promoter is described. The reaction occurs smoothly at room temperature under environmentally benign conditions without any catalyst, additive, ligand, or organic solvent. The developed sulfoxide synthetic protocol is attractive due to the use of water as the solvent and provides a novel and efficient route to a wide range of functionalized diaryl sulfoxides.

KW - indoles

KW - sulfinylation reaction

KW - trifluoroacetic acid

KW - water

UR - https://www.scopus.com/pages/publications/85107433557

U2 - 10.1134/S1070428021050109

DO - 10.1134/S1070428021050109

M3 - 文章

AN - SCOPUS:85107433557

SN - 1070-4280

VL - 57

SP - 831

EP - 841

JO - Russian Journal of Organic Chemistry

JF - Russian Journal of Organic Chemistry

IS - 5

ER -

Efficient Synthesis of 3-(Arenesulfinyl)indoles in Water

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Keywords

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